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MELK-IN-1

Product Specifications

CAS Number

2095596-44-2

Target

MELK

Related Pathways

PI3K/Akt/mTOR signaling

Purity

0.9984

Bioactivity

MELK-IN-1 (MELK inhibitor 17) is a potent inhibitor of maternal embryonic leucine zipper kinase (MELK), (IC50:3nm; Ki:0.39 nM) .

Smiles

COC(=O)c1ccc2NC(=O)\C(=C(/Nc3ccc(cc3)N(C)C(=O)CN3CCN(C)CC3)c3ccccc3)c2c1

Molecular Formula

C31H33N5O4

Molecular Weight

539.62

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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