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MARK4 inhibitor 1

Product Specifications

CAS Number

2271081-58-2

Target

Apoptosis, AMPK

Related Pathways

Chromatin/Epigenetic, Apoptosis, PI3K/Akt/mTOR signaling

Purity

0.9859

Bioactivity

MARK4 inhibitor 1 inhibits cancer cell proliferation, metastasis and induces apoptosis. MARK4 inhibitor 1 is a potent microtubule affinity-regulating kinase 4 (MARK4) inhibitor, with an IC50 of 1.54 μM.

Smiles

COc1ccc(Cn2cc(nn2)C(=O)N\N=C2\C(=O)Nc3c2cccc3C)cc1

Molecular Formula

C20H18N6O3

Molecular Weight

390.4

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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