MARK4 inhibitor 1
Product Specifications
CAS Number
2271081-58-2
Target
Apoptosis, AMPK
Related Pathways
Chromatin/Epigenetic, Apoptosis, PI3K/Akt/mTOR signaling
Purity
0.9859
Bioactivity
MARK4 inhibitor 1 inhibits cancer cell proliferation, metastasis and induces apoptosis. MARK4 inhibitor 1 is a potent microtubule affinity-regulating kinase 4 (MARK4) inhibitor, with an IC50 of 1.54 μM.
Smiles
COc1ccc(Cn2cc(nn2)C(=O)N\N=C2\C(=O)Nc3c2cccc3C)cc1
Molecular Formula
C20H18N6O3
Molecular Weight
390.4
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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