J-2156
Product Specifications
CAS Number
848647-56-3
Target
Others, Somatostatin
Related Pathways
Others, GPCR/G Protein
Bioactivity
The ED50 of J-2156 in rats for the relief of mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws was 3.7 and 8.0 mg/kg, respectively. J-2156 is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively.
Smiles
S(N[C@H](C(N[C@@H](CC1=CC=CC=C1)C(N)=O)=O)CCN)(=O)(=O)C=2C3=C(C(C)=CC2)C=CC=C3
Molecular Formula
C24H28N4O4S
Molecular Weight
468.57
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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