GSK3368715
Product Specifications
CAS Number
1629013-22-4
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Bioactivity
GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s: 3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8) ) . It has strong anti-cancer activity.
Smiles
C(OCC)C1(COCC)CCC(CC1)C=2C(CN(CCNC)C)=CNN2
Molecular Formula
C20H38N4O2
Molecular Weight
366.54
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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