Fiboflapon sodium
Product Specifications
CAS Number
1196070-26-4
Target
FLAP|||LTR|||Leukotriene Receptor
Related Pathways
Immunology/Inflammation|||GPCR/G Protein
Bioactivity
Fiboflapon sodium (GSK2190915) is an orally bioavailable 5-lipoxygenase-activating protein (FLAP) inhibitor with a potency of 2.9 nM in FLAP binding, an IC50 of 76 nM for inhibition of LTB4 in human blood.
Smiles
[Na].CCOc1ccc(cn1)-c1ccc(Cn2c(CC(C)(C)C(O)=O)c(SC(C)(C)C)c3cc(OCc4ccc(C)cn4)ccc23)cc1
Molecular Formula
C38H43N3NaO4S
Molecular Weight
660.83
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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