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GSK-5498A

Product Specifications

CAS Number

1253186-49-0

Target

Others, Calcium Channel

Related Pathways

Membrane transporter/Ion channel, Others, Metabolism

Bioactivity

GSK-5498A is a selective blocker of CARC (IC50, 1 μM) . It inhibits mediator release from mast cells, and pro-inflammatory cytokine release from T-cells in a variety of species.

Smiles

Fc1cccc(c1Cn1ccc(NC(=O)c2c(F)cccc2F)n1)C(F)(F)F

Molecular Formula

C18H11F6N3O

Molecular Weight

399.29

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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