GSK-5498A
Product Specifications
CAS Number
1253186-49-0
Target
Others, Calcium Channel
Related Pathways
Membrane transporter/Ion channel, Others, Metabolism
Bioactivity
GSK-5498A is a selective blocker of CARC (IC50, 1 μM) . It inhibits mediator release from mast cells, and pro-inflammatory cytokine release from T-cells in a variety of species.
Smiles
Fc1cccc(c1Cn1ccc(NC(=O)c2c(F)cccc2F)n1)C(F)(F)F
Molecular Formula
C18H11F6N3O
Molecular Weight
399.29
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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