Glucagon receptor antagonists-5
Product Specifications
CAS Number
2200274-63-9
Target
Others, Glucagon Receptor
Related Pathways
GPCR/G Protein, Others
Bioactivity
Glucagon receptor antagonists-5 is an orally bioavailable indazole-based glucagon receptor antagonist (Ki: 32 nM) . It has potential for the treatment of type 2 diabetes mellitus (T2DM) .
Smiles
[C@@H](CC(C)C)(N1C=2C(=CC(=C(C)C2)C3=C(Cl)C=C(C(F)(F)F)C=C3)C=N1)C4=CC=C(C(NCCC(O)=O)=O)C=C4
Molecular Formula
C30H29ClF3N3O3
Molecular Weight
572.02
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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