Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

GKI-1

Product Specifications

CAS Number

2444764-03-6

Target

ROCK, Others

Related Pathways

Stem Cells, Others, Cell Cycle/Checkpoint, Cytoskeletal Signaling

Purity

0.9996

Bioactivity

GKI-1 is a Greatwall (GWL) kinase inhibitor with an IC50 of 4.9 for hGWLFL and 2.5 μM for hGWL-KinDom. It exhibits stronger inhibition on ROCK1 with an IC50 of 11 μM and only weakly inhibits PKA.

Smiles

N(C=1C=C(C=CC1)C=2C=NNC2)C3=CC=C(Cl)C=C3

Molecular Formula

C15H12ClN3

Molecular Weight

269.73

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

DAPK3 siRNA (Rat)
CRR1887-01 15 nmol

DAPK3 siRNA (Rat)

Sign In for Pricing
View Details
DAPK3 siRNA (Rat)
CRR1887-02 30 nmol

DAPK3 siRNA (Rat)

Sign In for Pricing
View Details
GRK2 Antibody
orb69413 100 µL

GRK2 Antibody

Sign In for Pricing
View Details
Recombinant Rickettsia massiliae DNA replication and repair protein recF (recF)
MBS1262550-01 0.02 mg (E-Coli)

Recombinant Rickettsia massiliae DNA replication and repair protein recF (recF)

Sign In for Pricing
View Details
Recombinant Rickettsia massiliae DNA replication and repair protein recF (recF)
MBS1262550-02 0.02 mg (Yeast)

Recombinant Rickettsia massiliae DNA replication and repair protein recF (recF)

Sign In for Pricing
View Details
Recombinant Rickettsia massiliae DNA replication and repair protein recF (recF)
MBS1262550-03 0.1 mg (E-Coli)

Recombinant Rickettsia massiliae DNA replication and repair protein recF (recF)

Sign In for Pricing
View Details