What is the catalog number for GCN2-IN-6?

The catalog number for GCN2-IN-6 is T11374.

What sizes are available for GCN2-IN-6?

GCN2-IN-6 is available in the following size(s): 1 mg, 5 mg, 1 mL - 10 mM (in DMSO), 50 mg.

How many pack sizes does GCN2-IN-6 come in?

GCN2-IN-6 is available in 4 different pack sizes.

Is GCN2-IN-6 in stock?

GCN2-IN-6 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures GCN2-IN-6?

GCN2-IN-6 is manufactured by Molfinity.

What is the estimated delivery time for GCN2-IN-6?

Estimated delivery time for GCN2-IN-6 is approximately 10 business day(s), depending on your location.

GCN2-IN-6

Product Specifications

CAS Number

2183470-09-7

Target

PERK

Related Pathways

Apoptosis

Purity

0.98

Bioactivity

GCN2-IN-6 is a potent and orally available GCN2 inhibitor confirmed by in-house enzymatic (IC50: 1.8 nM) and cellular assays (IC50: 9.3 nM) . GCN2-IN-6 is also an eIF2α kinase PERK inhibitor with IC50s of 0.26 nM in enzymatic assay and 230 nM in cells respectively.