GB-110
Product Specifications
CAS Number
1252806-70-4
Target
Others, Protease-activated Receptor
Related Pathways
Others, GPCR/G Protein
Bioactivity
GB-110 selectively induces PAR2-mediated intracellular Ca2+ release in HT29 cells with an EC50 of 0.28 μM. GB-110 is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist.
Smiles
[C@H](CC1CCCCC1)(C(N[C@H](C(NCC2=CC(C(=O)N3CCC(CN)CC3)=CC=C2)=O)[C@H](CC)C)=O)NC(=O)C4=CC=NO4
Molecular Formula
C33H48N6O5
Molecular Weight
608.77
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
GTR15150074 1 Vial
Lentiviral mouse Car12 shRNA (UAS) - Lentiviral mouse Car12 shRNA (UAS, iRFP) (25)
Sign In for Pricing
View Details 
127612-HRP 100 µL
GSTO2 (Glutathione S-transferase omega-2, Glutathione S-transferase omega 2-2, Glutathione-dependent Dehydroascorbate Reductase, Monomethylarsonic Acid Reductase) (HRP)
Sign In for Pricing
View Details 
PB9661-Fluoro647 100 µg/Vial
Anti-LIFR Antibody Picoband® Fluoro647 Conjugated
Sign In for Pricing
View Details