Epertinib
Product Specifications
CAS Number
908305-13-5
Target
EGFR, HER
Related Pathways
JAK/STAT signaling, Tyrosine Kinase/Adaptors, Angiogenesis
Bioactivity
Epertinib is a reversible and selective tyrosine kinase inhibitor of EGFR, HER2, and HER4 (IC50s: 1.48 nM, 7.15 nM, and 2.49 nM) . It displays a strong antitumor activity.
Smiles
N(C=1C2=C(C=CC(\C(=N\OC[C@H]3COCCN3)\C#CC)=C2)N=CN1)C4=CC(Cl)=C(OCC5=CC(F)=CC=C5)C=C4
Molecular Formula
C30H27ClFN5O3
Molecular Weight
560.02
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
![Elab Fluor® Violet 450 Rat IgM, κ Isotype Control[RTK2118]](https://cdn.genprice.uk/products/763/68dd149b061270361e7cf064/imageurl/e-ab-f09773q.webp)
E-AB-F09773Q-01 25 µg
Elab Fluor® Violet 450 Rat IgM, κ Isotype Control[RTK2118]
Sign In for Pricing
View Details E-AB-F09773Q-02 100 µg
Elab Fluor® Violet 450 Rat IgM, κ Isotype Control[RTK2118]
Sign In for Pricing
View Details 
TRV-0004832-01 10 µg
Recombinant Inhibitor Of Nuclear Factor Kappa B Kinase Interacting Protein (IKBIP)
Sign In for Pricing
View Details TRV-0004832-02 50 µg
Recombinant Inhibitor Of Nuclear Factor Kappa B Kinase Interacting Protein (IKBIP)
Sign In for Pricing
View Details TRV-0004832-03 100 µg
Recombinant Inhibitor Of Nuclear Factor Kappa B Kinase Interacting Protein (IKBIP)
Sign In for Pricing
View Details