(R) -Elagolix
Product Specifications
CAS Number
834153-87-6
Target
GNRH Receptor
Related Pathways
GPCR/G Protein
Purity
0.9908
Bioactivity
(R) -Elagolix (NBI-56418) is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a dose-dependent suppression of ovarian estrogen production, that is, from partial suppression at lower doses to full suppression at higher doses.
Smiles
[H][C@@](Cn1c(=O)c(c(C)n(Cc2c(F)cccc2C(F)(F)F)c1=O)-c1cccc(OC)c1F)(NCCCC(O)=O)c1ccccc1
Molecular Formula
C32H30F5N3O5
Molecular Weight
631.59
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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