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DRAK2-IN-1

Product Specifications

CAS Number

871837-60-4

Target

Others, DAPK

Related Pathways

Apoptosis, Others

Bioactivity

Drak2-in-1, a potent, selective and ATP-competitive DRAK2 inhibitor, has an IC50 and KIvalue of 3 nM and 0.26 nM, respectively.Drak2-in-1 also had an effect on DRAK1 (IC50=51 nM) .

Smiles

CCCCC(=O)Nc1ccc2NC(=O)\C(=C3/Nc4ccccc4/C/3=N/O)c2c1

Molecular Formula

C21H20N4O3

Molecular Weight

376.41

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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