What is the catalog number for Samuraciclib hydrochloride?

The catalog number for Samuraciclib hydrochloride is T10898.

What sizes are available for Samuraciclib hydrochloride?

Samuraciclib hydrochloride is available in the following size(s): 1 mg, 2 mg, 5 mg, 1 mL - 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg.

How many pack sizes does Samuraciclib hydrochloride come in?

Samuraciclib hydrochloride is available in 8 different pack sizes.

Is Samuraciclib hydrochloride in stock?

Samuraciclib hydrochloride is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Samuraciclib hydrochloride?

Samuraciclib hydrochloride is manufactured by Molfinity.

What is the estimated delivery time for Samuraciclib hydrochloride?

Estimated delivery time for Samuraciclib hydrochloride is approximately 10 business day(s), depending on your location.

Samuraciclib hydrochloride

Product Specifications

CAS Number

1805789-54-1

Target

Apoptosis, CDK

Related Pathways

Cell Cycle/Checkpoint, Apoptosis

Purity

0.998

Bioactivity

Samuraciclib hydrochloride (ICEC0942 hydrochloride) is a potent, selective, ATP competitive and oral active CDK7 inhibitor with IC50 of 41 nM. The selectivity of Samuraciclib hydrochloride is 45-, 15-, 230- and 30-fold higher than CDK1, CDK2 (IC50 is 578 nM), CDK5 and CDK9 respectively. Samuraciclib hydrochloride inhibits the growth of breast cancer cell lines with GI50 values between 0.2-0.3 μM. Samuraciclib hydrochloride has anti-tumor effects.