Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

CSRM617 hydrochloride

Product Specifications

CAS Number

1353749-74-2

Target

Apoptosis, Androgen Receptor

Related Pathways

Apoptosis, Endocrinology/Hormones

Purity

0.9959

Bioactivity

CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 (OC2, a master regulator of androgen receptor), with a Kd of 7.43 μM in SPR assays, directly binding to the OC2-HOX domain. CSRM617 hydrochloride induces apoptosis through the appearance of cleaved Caspase-3 and PARP and is well tolerated in the mouse model of prostate cancer [1].

Smiles

Cl.NC(CO)C(=O)N\N=C\c1ccc(O)c(O)c1O

Molecular Formula

C10H14ClN3O5

Molecular Weight

291.69

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Mouse Acadm/Medium-chain specific acyl-CoA dehydrogenase, mitochondrial ELISA Kit
orb1661998 96 Tests

Mouse Acadm/Medium-chain specific acyl-CoA dehydrogenase, mitochondrial ELISA Kit

Sign In for Pricing
View Details
N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide
WWC91178-01 10 mg

N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide

Sign In for Pricing
View Details
N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide
WWC91178-02 25 mg

N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide

Sign In for Pricing
View Details
N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide
WWC91178-03 50 mg

N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide

Sign In for Pricing
View Details
N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide
WWC91178-04 100 mg

N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide

Sign In for Pricing
View Details
N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide
WWC91178-05 250 mg

N- (2,5-diaza-2- (2- (2-bromophenyl) -2-oxoethyl) -3-oxo-6-phenylbicyclo[5.4.0]undeca-1 (11),5,7 (8),9-tetraen-4-yl) -2- (3-methoxyphenyl) eth anamide

Sign In for Pricing
View Details