Gartisertib
Product Specifications
CAS Number
1613191-99-3
Target
ATM/ATR
Related Pathways
PI3K/Akt/mTOR signaling, DNA Damage/DNA Repair
Purity
0.9952
Bioactivity
Gartisertib (VX-803) is an orally active and selective Rad3-related protein (ATR) inhibitor with antitumor activity, inhibiting the antiproliferative effect induced in ccRCC cells, and inhibiting ATR-driven phosphorylation of checkpoint kinase 1 (Chk1), useful for studying solid tumors.
Smiles
O=C(NC=1C=NC=C(F)C1N2CCC(C(=O)N3CCN(CC3)C4COC4)CC2)C=5C(=NN6C=C(F)C=NC56)N
Molecular Formula
C25H29F2N9O3
Molecular Weight
541.55
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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