Gartisertib
Product Specifications
CAS Number
1613191-99-3
Target
ATM/ATR
Related Pathways
PI3K/Akt/mTOR signaling|||DNA Damage/DNA Repair
Purity
0.9952
Bioactivity
Gartisertib (VX-803) is an orally active and selective Rad3-related protein (ATR) inhibitor with antitumor activity, inhibiting the antiproliferative effect induced in ccRCC cells, and inhibiting ATR-driven phosphorylation of checkpoint kinase 1 (Chk1), useful for studying solid tumors.
Smiles
O=C(NC=1C=NC=C(F)C1N2CCC(C(=O)N3CCN(CC3)C4COC4)CC2)C=5C(=NN6C=C(F)C=NC56)N
Molecular Formula
C25H29F2N9O3
Molecular Weight
541.55
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
TL519372V 500 µL Each
1700016C15Rik Mouse shRNA Lentiviral Particle (Locus ID 69428)
Ask
View Details 
MBS6397755-01 0.1 mL
TYRO3 (Tyrosine-protein Kinase Receptor TYRO3, Tyrosine-protein Kinase BYK, BYK, Tyrosine-protein Kinase DTK, DTK, Tyrosine-protein Kinase RSE, RSE, Tyrosine-protein Kinase SKY, SKY, Tyrosine-protein Kinase TIF, TIF) APC
Ask
View Details MBS6397755-02 5x 0.1 mL
TYRO3 (Tyrosine-protein Kinase Receptor TYRO3, Tyrosine-protein Kinase BYK, BYK, Tyrosine-protein Kinase DTK, DTK, Tyrosine-protein Kinase RSE, RSE, Tyrosine-protein Kinase SKY, SKY, Tyrosine-protein Kinase TIF, TIF) APC
Ask
View Details