AS2717638
Product Specifications
CAS Number
2148339-28-8
Target
Others, LPL Receptor
Related Pathways
Others, GPCR/G Protein
Purity
0.9923
Bioactivity
AS2717638 is an orally active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist (IC50: 38 nM for hLPA5) . It also significantly improves PGF2α-, PGE2-, and AMPA-induced allodynia.
Smiles
COc1cc2c(cn(-c3noc4ccc(C)cc34)c(=O)c2cc1OC)C(=O)N1CCCCC1
Molecular Formula
C25H25N3O5
Molecular Weight
447.48
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog