AR-A 2
Product Specifications
CAS Number
220051-79-6
Target
Others|||5-HT Receptor
Related Pathways
GPCR/G Protein|||Neuroscience|||Others
Bioactivity
AR-A 2 is a selective 5-HT1B receptor antagonist with high affinity to guinea pig cortex 5-HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0.47 nM), exhibiting a 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki: 5 nM) .
Smiles
CC1=C2C(=C(C=C1)N3CCN(C)CC3)C[C@H](NC(=O)C4=CC=C(C=C4)N5CCOCC5)CC2
Molecular Formula
C27H36N4O2
Molecular Weight
448.6
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
