Aprocitentan D4

Product Specifications

Bioactivity

Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is a dual ETA/ETB antagonist (IC50s: 3.4 nM and 987 nM; pA2s: 6.7 and 5.5) .

Smiles

O=S(N)(NC1=NC=NC(OC([2H])([2H])C([2H])([2H])OC2=NC=C(Br)C=N2)=C1C3=CC=C(Br)C=C3)=O

Molecular Formula

C16H10D4Br2N6O4S

Molecular Weight

550.22

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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