(5Z,2E) -CU-3
Product Specifications
CAS Number
1815598-71-0
Target
Apoptosis
Related Pathways
Apoptosis
Purity
0.9902
Bioactivity
(5Z,2E) -CU-3 is a potent and highly selective inhibitor of the DGK? isozyme with an IC50 value of 0.6 ?M, competing with ATP and exhibiting a Km value of 0.48 mM. It specifically targets the catalytic region of DGK? without affecting the regulatory region and has demonstrated antitumor and immunogenic effects by promoting cancer cell apoptosis and T cell activation.
Smiles
O=C1N(NS(=O)(=O)c2ccccc2)C(=S)S\C1=C/C=C/c1ccco1
Molecular Formula
C16H12N2O4S3
Molecular Weight
392.47
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
MBS6288857-01 0.2 mL
CRISPLD2, NT (CRISPLD2, CRISP11, LCRISP2, Cysteine-rich secretory protein LCCL domain-containing 2, Cysteine-rich secretory protein 11, LCCL domain-containing cysteine-rich secretory protein 2) (AP)
Ask
View Details MBS6288857-02 5x 0.2 mL
CRISPLD2, NT (CRISPLD2, CRISP11, LCRISP2, Cysteine-rich secretory protein LCCL domain-containing 2, Cysteine-rich secretory protein 11, LCCL domain-containing cysteine-rich secretory protein 2) (AP)
Ask
View Details