Pitofenone hydrochloride
Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively[1][2].
Product Specifications
CAS Number
1248-42-6
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335, H360
Target
Cholinesterase (ChE)
Type
Reference compound
Related Pathways
Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Pitofenone_hydrochloride.html
Purity
99.88
Solubility
DMSO : 83.33 mg/mL (ultrasonic) |H2O : 100 mg/mL (ultrasonic)
Smiles
Cl[H].O=C(C1=CC=C(C=C1)OCCN2CCCCC2)C3=C(C=CC=C3)C(OC)=O
Molecular Formula
C22H26ClNO4
Molecular Weight
403.90
Precautions
H302, H315, H319, H335, H360
References & Citations
[1]Punekar NS, et al. Acetylcholinesterase inhibition by pitofenone: a spasmolytic compound. Biotechnol Appl Biochem. 1991 Dec;14 (3) :378-82.|[2]https://journals.lww.com/iphr/abstract/1998/30050/antispasmodic_activity_of_diclofenac_and_its.6.aspx
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
AChE
Available Sizes
Frequently Asked Questions
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