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TC-S 7010

TC-S 7010 is a potent and selective inhibitor of Aurora kinase A (IC₅₀ = 3.4 nM). It displays1000-fold selectivity for Aurora kinase A over Aurora kinase B. Displays antiproliferative activity in HCT116 and HT29 cells (IC₅₀ values are 0.19 and 2.9 μM respectively).

Product Specifications

Shipping Conditions

gel pack

Storage Conditions

-20°C

Shelf Life

36 months

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