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ZSTK474

ZSTK474 is a reversible, potent and specific inhibitor of phosphoinositide 3-kinase (PI3K) isoforms ((IC₅₀s = 17, 53, and 6 nM for p110β, -γ, and -δ, respectively). More effective than LY 294,002 in vitro and as in vivo. Displays strong antitumor activities against human cancer xenografts (A549, PC-3 and WiDr) when administered orally to mice.

Product Specifications

Shipping Conditions

Gel Pack

Storage Conditions

-20°C

Shelf Life

36 months

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MBS1481766-04 0.1 mg (Yeast)

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MBS1481766-06 0.02 mg (Mammalian-Cell)

Recombinant Streptomyces avermitilis NADH-quinone oxidoreductase subunit B 1 (nuoB1)

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