Transcription factor-IN-1
Transcription factor-IN-1 (Compound 4e) is an inhibitor for transcription factor. Transcription factor-IN-1 exhibits anticonvulsant activity by antagonism with pentylenetetrazole (PTZ) (ED50 =34.5 mg/kg) . Transcription factor-IN-1 exhibits antidepressant effects in rat models[1].
Product Specifications
UNSPSC
12352005
Target
GABA Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/transcription-factor-in-1.html
Smiles
O=C(OCC)C1=C(SCC(NC(C2=CC=CC=C2)C3=CC=CC=C3)=O)N=C(N4CCCC4)C=C1C5=CC=CC=C5
Molecular Formula
C33H33N3O3S
Molecular Weight
551.70
References & Citations
[1]Sh Dashyan S, et al., Synthesis, evaluation of biological activity and SAR of new thioalkyl derivatives of pyridine. Bioorg Chem. 2024 Jul;148:107435.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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