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TG 100713

Product Specifications

UNSPSC Description

TG 100713 is an inhibitor of PI3K, with IC50s of 24, 50, 165, and 215 nM for PI3Kδ, γ, α and β isoforms respectively[1].

Target Antigen

PI3K

Type

Reference compound

Related Pathways

PI3K/Akt/mTOR

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/tg-100713.html

Smiles

OC1=CC=CC(C2=NC3=C(N)N=C(N)N=C3N=C2)=C1

Molecular Weight

254.25

References & Citations

[1]Doukas J, et, al. Phosphoinositide 3-kinase gamma/delta inhibition limits infarct size after myocardial ischemia/reperfusion injury. Proc Natl Acad Sci U S A. 2006 Dec 26;103(52):19866-71.

Shipping Conditions

Room Temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-13514/TG-100713-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-13514/TG-100713-SDS-MedChemExpress.pdf

CAS Number

925705-73-3

Available Sizes

Curated Selection

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