TG 100713
Product Specifications
UNSPSC Description
TG 100713 is an inhibitor of PI3K, with IC50s of 24, 50, 165, and 215 nM for PI3Kδ, γ, α and β isoforms respectively[1].
Target Antigen
PI3K
Type
Reference compound
Related Pathways
PI3K/Akt/mTOR
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/tg-100713.html
Smiles
OC1=CC=CC(C2=NC3=C(N)N=C(N)N=C3N=C2)=C1
Molecular Weight
254.25
References & Citations
[1]Doukas J, et, al. Phosphoinositide 3-kinase gamma/delta inhibition limits infarct size after myocardial ischemia/reperfusion injury. Proc Natl Acad Sci U S A. 2006 Dec 26;103(52):19866-71.
Shipping Conditions
Room Temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-13514/TG-100713-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-13514/TG-100713-SDS-MedChemExpress.pdf
CAS Number
925705-73-3
Available Sizes
Curated Selection
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