MSK-195
MSK-195 is a potent agonist of TRPV1, with a potency of 120 nM and an efficacy of 71% in arteriolar response[1].
Product Specifications
CAS Number
289902-82-5
UNSPSC
12352005
Target
TRP Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/msk-195.html
Smiles
CC(C)(C(OCC(CNC(CC1=CC=C(C(OC)=C1)OCCN)=O)CC2=CC=C(C(C)=C2)C)=O)C
Molecular Formula
C28H40N2O5
Molecular Weight
484.63
References & Citations
[1]Á Czikora, et al. Structure-activity relationships of vanilloid receptor agonists for arteriolar TRPV1. Br J Pharmacol. 2012 Mar; 165 (6) : 1801–1812.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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