MS0124
MS0124 is a potent selective G9a-like protein (GLP) inhibitor with IC50 values of 13±4 nM and 440±63 nM for GLP and G9a, respectively[1].
Product Specifications
CAS Number
[1197196-63-6]
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ms0124.html
Purity
99.79
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
CN(CC1)CCC1NC(N=C(N2CCOCC2)N=C3C=C4OC)=C3C=C4OC
Molecular Formula
C20H29N5O3
Molecular Weight
387.48
References & Citations
[1]Yan Xiong, et al. Structure-activity relationship studies of G9a-like protein (GLP) inhibitors. Bioorg Med Chem
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
EHMT1/GLP/KMT1D; EHMT2/G9a/KMT1C
Available Sizes
Curated Selection
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