PSB-SB-1203
PSB-SB-1203 (Compound 25b) is a dual CB1/CB2 ligand that blocks CB1 but activates CB2 receptors (CB1 Ki 0.244 μM; CB2 Ki 0.210 μM, EC50 0.054 μM) . PSB-SB-1203 is promising for research of obesity and cancers[1].
Product Specifications
CAS Number
[1399049-80-9]
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Cancer; Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/psb-sb-1203.html
Smiles
O=C1OC2=C(C=C1CC3=C(O)C=CC=C3)C(O)=CC(C(C)(CCCCCC)C)=C2
Molecular Formula
C25H30O4
Molecular Weight
394.50
References & Citations
[1]Rempel V, et al. 7-Alkyl-3-benzylcoumarins: a versatile scaffold for the development of potent and selective cannabinoid receptor agonists and antagonists. J Med Chem. 2012 Sep 27;55 (18) :7967-77.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CB1; CB2
Curated Selection
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