RL5a
RL5a (compund C23) is a SETD8 inhibitor[1].
Product Specifications
CAS Number
[133671-66-6]
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/rl5a.html
Purity
99.6
Solubility
DMSO : 40 mg/mL (ultrasonic; warming)
Smiles
CN(C)CCNC1=CC(C2=CC=CO2)=NC3=CC=CC=C13
Molecular Formula
C17H19N3O
Molecular Weight
281.35
References & Citations
[1]Gardner NJ, et al. The High-Affinity Interaction between ORC and DNA that Is Required for Replication Licensing Is Inhibited by 2-Arylquinolin-4-Amines. Cell Chem Biol. 2017 Aug 17;24 (8) :981-992.e4.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
