Morphiceptin

Morphiceptin is a potent and specific agonist for morphine (μ) receptors. Morphiceptin, as a synthetic peptide, is the amide of a fragment of the milk protein β-casein. Morphiceptin has morphinelike activities and is highly specific for morphine (μ) receptors but not for Enkephalin receptors[1].

Product Specifications

CAS Number

[74135-04-9]

UNSPSC

12352209

Target

Opioid Receptor

Type

Peptides

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease; Cardiovascular Disease

Assay Protocol

https://www.medchemexpress.com/morphiceptin.html

Purity

99.07

Solubility

DMSO : 100 mg/mL (ultrasonic) |H2O : ≥ 250 mg/mL

Smiles

O=C([C@H]1N(CCC1)C([C@@H](NC([C@H]2N(CCC2)C([C@@H](N)CC3=CC=C(C=C3)O)=O)=O)CC4=CC=CC=C4)=O)N

Molecular Formula

C28H35N5O5

Molecular Weight

521.61

References & Citations

[1]Chang KJ, et al. Morphiceptin (NH4-tyr-pro-phe-pro-COHN2) : a potent and specific agonist for morphine (mu) receptors. Science. 1981;212 (4490) :75-77.