11β-HSD1-IN-1

11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1), with an IC50 of 52 nM, and used for the treatment of pain.

Product Specifications

CAS Number

[1203956-47-1]

UNSPSC

12352005

Target

11β-HSD

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/4H-1,2,4-Triazole,_3-_2-chloro-4-fluorophenyl_-4-methyl-5-[1-methyl-1-_2,4,6-trifluorophenoxy_ethyl]-.html

Purity

99.80

Solubility

10 mM in DMSO

Smiles

CC(C1=NN=C(C2=CC=C(F)C=C2Cl)N1C)(C)OC3=C(F)C=C(F)C=C3F

Molecular Formula

C18H14ClF4N3O

Molecular Weight

399.77

References & Citations

[1]THERAPEUTIC AGENT FOR PAIN. WO2012033070A1

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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