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GFH018

GFH018 is a TGF-βRI inhibitor. GFH018 can be used for cancer research[1].

Product Specifications

CAS Number

[2169299-67-4]

UNSPSC

12352005

Target

TGF-β Receptor

Type

Reference compound

Related Pathways

TGF-beta/Smad

Applications

Cancer-Kinase/protease

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/tgf-βri-inhibitor-1.html

Purity

98.27

Solubility

10 mM in DMSO

Smiles

NC(/C=C/C1=C(C=CC2=NC=NN21)C3=C(CCC4)N4N=C3C5=CC=CC(C)=N5)=O

Molecular Formula

C21H19N7O

Molecular Weight

385.42

References & Citations

[1]Wu, et al. Crystal form and salt form of TGF- β RI inhibitor and preparation method thereof. Patent, CN111479809A.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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