Adenosine receptor antagonist 1
Product Specifications
UNSPSC Description
Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aR than A2bR.
Target Antigen
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/adenosine-receptor-antagonist-1.html
Solubility
10 mM in DMSO
Smiles
NC1=NC(C2=CC=CC=C2)=C(C3=NC(CC4=C(C=C(C=N4)F)Cl)=NN13)C5=CNC(C=C5)=O
Molecular Weight
447.85
References & Citations
[1]Lamb ML, et al. Triazole compounds as adenosine receptor antagonists. WO2021156439A1.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-141865/Adenosine-receptor-antagonist-1-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-141865/
Clinical Information
No Development Reported
CAS Number
2682930-40-9
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