Adenosine receptor antagonist 1
Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aR than A2bR.
Product Specifications
CAS Number
[2682930-40-9]
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/adenosine-receptor-antagonist-1.html
Solubility
10 mM in DMSO
Smiles
NC1=NC(C2=CC=CC=C2)=C(C3=NC(CC4=C(C=C(C=N4)F)Cl)=NN13)C5=CNC(C=C5)=O
Molecular Formula
C22H15ClFN7O
Molecular Weight
447.85
References & Citations
[1]Lamb ML, et al. Triazole compounds as adenosine receptor antagonists. WO2021156439A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
Adenosine A2A receptor (A2AR)
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