Adenosine receptor antagonist 1
Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aR than A2bR.
Product Specifications
CAS Number
[2682930-40-9]
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/adenosine-receptor-antagonist-1.html
Solubility
10 mM in DMSO
Smiles
NC1=NC(C2=CC=CC=C2)=C(C3=NC(CC4=C(C=C(C=N4)F)Cl)=NN13)C5=CNC(C=C5)=O
Molecular Formula
C22H15ClFN7O
Molecular Weight
447.85
References & Citations
[1]Lamb ML, et al. Triazole compounds as adenosine receptor antagonists. WO2021156439A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
Adenosine A2A receptor (A2AR)
Curated Selection
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