VPC13163
VPC13163 is a potent androgen receptor (AR) BF3 inhibitor with an IC50 of 0.31 µM. VPC13163 has anticancer effects[1].
Product Specifications
CAS Number
[6637-10-1]
UNSPSC
12352005
Hazard Statement
H302, H317
Target
Androgen Receptor
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/vpc13163.html
Solubility
10 mM in DMSO
Smiles
C1(NC2=C(C1)C=CC=C2)C3=CNC4=C3C=CC=C4
Molecular Formula
C16H14N2
Molecular Weight
234.30
Precautions
H302, H317
References & Citations
[1]Ravi Shashi Nayana Munuganti, et al. Abstract 2508: The development of anti-androgens with a novel mechanism of action for treatment of castration-resistant prostate cancer. Cancer Res (2014) 74 (19_Supplement) : 2508.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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