GV-150013

GV-150013 is a selective CCK-B receptor antagonist. GV-150013 has sleep aid effect[1].

Product Specifications

CAS Number

[167355-22-8]

UNSPSC

12352005

Target

Cholecystokinin Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Field of Research

Others

Assay Protocol

https://www.medchemexpress.com/gv-150013.html

Solubility

10 mM in DMSO

Smiles

O=C([C@@H](C1=O)NC(NC2=CC=CC=C2)=O)N(C3=CC=CC=C3)C4=CC=CC=C4N1CC56CC7CC(CC(C7)C6)C5

Molecular Formula

C33H34N4O3

Molecular Weight

534.65

References & Citations

[1]Crespi F. Cholecystokinin-B (CCK-B) receptor antagonists improve "aged" sleep: a new class of sleep modulators? Methods Find Exp Clin Pharmacol. 1999 Jan-Feb;21 (1) :31-8.|[2]F.Crespi, et al. Influence of cholecystokinin-B (CCK-B) receptor antagonists on rat electroencephalography (EEG) : A new class of sleep modulators? Gaviraghi. Dept of Pharmacology GlaxoWellcome S.p.A., Medicine Research Centre, via A. Fleming, 4, 37135 Verona, Italy