Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Lusaperidone

Product Specifications

UNSPSC Description

Lusaperidone (R107474) is an α2 adrenergic receptor antagonist with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively.

Target Antigen

Adrenergic Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein;Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease; Endocrinology

Assay Protocol

https://www.medchemexpress.com/Lusaperidone.html

Purity

99.81

Solubility

DMSO : 3.45 mg/mL (ultrasonic;warming;heat to 60°C)

Smiles

O=C1C(CCN2CCC(OC3=CC=CC=C34)=C4C2)=C(C)N=C5N1C=CC=C5

Molecular Weight

359.42

References & Citations

[1]Van der Mey M, et al. Synthesis and biodistribution of [11C]R107474, a new radiolabeled alpha2-adrenoceptor antagonist. Bioorg Med Chem. 2006 Jul 1;14(13):4526-34.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-U00117/Lusaperidone-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-U00117/Lusaperidone-SDS-MedChemExpress.pdf

Clinical Information

No Development Reported

CAS Number

214548-46-6

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

AK1 (Adenylate Kinase 1) (MaxLight 650)
MBS6226450-01 0.1 mL

AK1 (Adenylate Kinase 1) (MaxLight 650)

Ask
View Details
AK1 (Adenylate Kinase 1) (MaxLight 650)
MBS6226450-02 5x 0.1 mL

AK1 (Adenylate Kinase 1) (MaxLight 650)

Ask
View Details
Recombinant Escherichia coli UPF0265 protein yeeX (yeeX)
MBS1168575-01 0.02 mg (E-Coli)

Recombinant Escherichia coli UPF0265 protein yeeX (yeeX)

Ask
View Details
Recombinant Escherichia coli UPF0265 protein yeeX (yeeX)
MBS1168575-02 0.1 mg (E-Coli)

Recombinant Escherichia coli UPF0265 protein yeeX (yeeX)

Ask
View Details
Recombinant Escherichia coli UPF0265 protein yeeX (yeeX)
MBS1168575-03 0.02 mg (Yeast)

Recombinant Escherichia coli UPF0265 protein yeeX (yeeX)

Ask
View Details
Recombinant Escherichia coli UPF0265 protein yeeX (yeeX)
MBS1168575-04 0.1 mg (Yeast)

Recombinant Escherichia coli UPF0265 protein yeeX (yeeX)

Ask
View Details