Enrasentan
Product Specifications
UNSPSC Description
Enrasentan (SB 217242) is an endothelin (ET) receptor antagonist. Enrasentan has antihypertensive effects[1].
Target Antigen
Endothelin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/enrasentan.html
Smiles
O=C(O)[C@@H]1[C@H](C2=C([C@H]1C3=CC=C(C=C3OCCO)OC)C=C(C=C2)OCCC)C4=CC5=C(C=C4)OCO5
Molecular Weight
506.54
References & Citations
[1]Alessandro Cosenzi, et al. Antihypertensive treatment with enrasentan (SB217242) in an animal model of hypertension and hyperinsulinemia. J Cardiovasc Pharmacol. 2002 Apr;39(4):488-95.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-119667/Enrasentan-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-119667/
Clinical Information
Phase 2
CAS Number
167256-08-8
Curated Selection
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