Chalepensin
Chalepensin, a furanocoumarin, is a competitive CYP2A6 inhibitor. Chalepensin also inhibits human CYP1A1, CYP1A2, CYP2A13, CYP2C9, CYP2D6, CYP2E1, and CYP3A4 to different extents[1].
Product Specifications
CAS Number
[13164-03-9]
UNSPSC
12352005
Target
Cytochrome P450
Type
Natural Products
Related Pathways
Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/chalepensin.html
Purity
98.0
Solubility
10 mM in DMSO
Smiles
O=C1C(C(C)(C)C=C)=CC2=CC3=C(OC=C3)C=C2O1
Molecular Formula
C16H14O3
Molecular Weight
254.28
References & Citations
[1]Yune-Fang Ueng, et al. Mechanism-based inhibition of CYP1A1 and CYP3A4 by the furanocoumarin chalepensin. Drug Metab Pharmacokinet. 2013;28 (3) :229-38.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C (Powder, protect from light)
Scientific Category
Natural Products
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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