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MPX-007

Product Specifications

UNSPSC Description

MPX-007 is a GluN2A antagonist (IC50: 27 nM). MPX-007 is a tools to probe GluN2A physiology, and to study neuropsychiatric and developmental disorders[1].

Target Antigen

iGluR

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel;Neuronal Signaling

Applications

Neuroscience-Neurodegeneration

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/mpx-007.html

Solubility

10 mM in DMSO

Smiles

O=C(NCC1=CN=C(S1)C)C2=NC(C)=C(N=C2)CNS(=O)(C3=CC=C(C(F)=C3)F)=O

Molecular Weight

453.49

References & Citations

[1]Volkmann RA, et al. MPX-004 and MPX-007: New Pharmacological Tools to Study the Physiology of NMDA Receptors Containing the GluN2A Subunit. PLoS One. 2016 Feb 1;11(2):e0148129.

Shipping Conditions

Room temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-116483/MPX-007-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-116483/

Clinical Information

No Development Reported

CAS Number

1688685-29-1

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