Endomorphin 2 (TFA)
Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].
Product Specifications
CAS Number
[1276124-00-5]
UNSPSC
12352209
Target
Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/endomorphin-2-tfa.html
Purity
99.04
Solubility
DMSO : < 1 mg/mL|H2O : 125 mg/mL (ultrasonic)
Smiles
O=C(N)[C@H](CC1=CC=CC=C1)NC([C@H](CC2=CC=CC=C2)NC([C@H]3N(C([C@H](CC4=CC=C(C=C4)O)N)=O)CCC3)=O)=O.OC(C(F)(F)F)=O
Molecular Formula
C34H38F3N5O7
Molecular Weight
685.69
References & Citations
Shipping Conditions
Blue Ice
Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
μ Opioid Receptor/MOR
Available Sizes
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