CB1 antagonist 5
Product Specifications
UNSPSC Description
CB1 antagonist 5 (Compound 25) is an antagonist for CB1 cannabinoid receptor, with a Ki of 243 nM and an EC50 of 195 nM[1].
Target Antigen
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cb1-antagonist-5.html
Smiles
O=C1N(C(C(N1C2=CC=C(C=C2)Br)C3=CC=CC=C3)=O)C4=CC=C(C=C4)Br
Molecular Weight
486.16
References & Citations
[1]Muccioli GG, et al., Synthesis and activity of 1,3,5-triphenylimidazolidine-2,4-diones and 1,3,5-triphenyl-2-thioxoimidazolidin-4-ones: characterization of new CB1 cannabinoid receptor inverse agonists/antagonists. J Med Chem. 2006 Feb 9;49(3):872-82.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-120653/CB1-antagonist-5-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-120653/
Clinical Information
No Development Reported
CAS Number
878533-35-8
Curated Selection
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