Poneratoxin (acetate)

Poneratoxin acetate is the acetate salt form of Poneratoxin (HY-P10234) . Poneratoxin acetate is the modulator for voltage-gated sodium channel (NaV, EC50 for NaV1.6 and NaV1.7 is 97 nM and 2.3 µM), that lowers the voltage threshold for activation and inhibits the inactivation of channels, enhances the excitability of neurons, and leads to the transmission of pain signals[1].

Product Specifications

UNSPSC

12352209

Target

Sodium Channel

Related Pathways

Membrane Transporter/Ion Channel

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Purity

98.77

Solubility

DMSO : 125 mg/mL (ultrasonic)

Smiles

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