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PROTAC HPK1 Degrader-6

PROTAC HPK1 Degrader-6 is a highly efficient and effective PROTAC degrader targeting HPK1 (IC50 [1].

Product Specifications

CAS Number

[3099168-12-1]

UNSPSC

12352005

Target

MAP4K; PROTACs

Related Pathways

MAPK/ERK Pathway; PROTAC

Field of Research

Cancer

Smiles

O=C(N1)N(C2=CC=C(C3CCN(C4CN(C5=CC=C(NC6=NC=C7C=CC(C8=CN=C9OCCNC9=C8C)=CC7=N6)C=C5)C4)CC3)C=C2C)CCC1=O

Molecular Formula

C41H43N9O3

Molecular Weight

709.84

References & Citations

[1]Preparation of quinazoline heterobifunctional compounds for the degradation of HPK1, WO2025163390, Toure.

Shipping Conditions

Room temperature

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-178459/

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Curated Selection

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