Tanerasertib
Tanerasertib (Compound 456) is an AKT1 inhibitor with an IC50 of less than 15 nM against AKT1 E17K. Tanerasertib can be used in the study of cancer[1].
Product Specifications
CAS Number
[3034255-93-8]
UNSPSC
12352005
Target
Akt
Related Pathways
PI3K/Akt/mTOR
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Purity
98.87
Solubility
DMSO : 10 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
N#CC1=NC=CC(NC2CCN(CC2)CC3=CC=C(N4C5=C(N=C4C6=CC=CN=C6N)C=CC(C7=CC=C(F)C=N7)=N5)C=C3)=N1
Molecular Formula
C33H28FN11
Molecular Weight
597.65
References & Citations
[1]Michael David Bartberger, et al. Akt1 modulators. WO2024073371A1. 2024-04-04.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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