MU1920
MU1920 is an ATP-competitive, selective inhibitor for haspin with an IC50 of 6 nM. MU1920 exhibits good pharmacokinetic properties and metabolic stability in mouse plasma and microsomes without obvious anticancer effects, which can be used for development of chemical probes[1].
Product Specifications
CAS Number
[3067968-52-6]
UNSPSC
12352005
Target
Haspin Kinase
Related Pathways
Cell Cycle/DNA Damage
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Smiles
CN1N=C(NC2=CC=C(SC=C3C4=CC=NC=C4)C3=N2)C(C)=C1
Molecular Formula
C17H15N5S
Molecular Weight
321.40
References & Citations
[1]Moyano PM, et al., Thieno[3,2-b]pyridine: Attractive scaffold for highly selective inhibitors of underexplored protein kinases with variable binding mode. Angew Chem Int Ed Engl. 2025 Jan 2;64 (1) :e202412786.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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