PAR-2-IN-2
PAR-2-IN-2 (compound P-596) is a protease-activated receptor 2 (PAR-2) inhibitor with an IC50 of 10.79 μM for SLIGKV and an IC50 of greater than 200 μM for Trypsin[1].
Product Specifications
CAS Number
[313986-65-1]
UNSPSC
12352005
Target
Protease Activated Receptor (PAR) ; Ser/Thr Protease
Related Pathways
GPCR/G Protein; Metabolic Enzyme/Protease
Field of Research
Inflammation/Immunology
Smiles
O=C(N1CCN(CC1)C(C2=CC=CC=C2)=O)C3=NN4C(N=C(C5=CC=CC=C5)C=C4C(F)(F)F)=C3
Molecular Formula
C25H20F3N5O2
Molecular Weight
479.45
References & Citations
[1]Luc J. Farmer, et al. Imidazopyridazines useful as inhibitors of the par-2 signaling pathway. WO. WO2015048245 A1. 2014-09-25.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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