CP 524515

CP 524515 is a potent inhbitor of cholesteryl ester transfer protein (CETP) that leads to elevated high-density lipoprotein cholesterol levels[1].

Product Specifications

CAS Number

[262352-13-6]

UNSPSC

12352005

Target

CETP

Related Pathways

Metabolic Enzyme/Protease

Field of Research

Metabolic Disease

Smiles

FC(F)(F)C1=CC(C(F)(F)F)=CC(CN([C@@H]2C3=CC(C(F)(F)F)=CC=C3N([C@@H](C2)CC)C(OC(C)C)=O)C(OC)=O)=C1

Molecular Formula

C27H27F9N2O4

Molecular Weight

614.50

References & Citations

[1]Natalie L Trevaskis, et al. The Mechanism of Lymphatic Access of Two Cholesteryl Ester Transfer Protein Inhibitors (CP524,515 and CP532,623) and Evaluation of Their Impact on Lymph Lipoprotein Profiles. Pharm Res. 2010 Sep;27 (9) :1949-64. doi: 10.1007/s11095-010-0199-2.